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 | mAChRsTooltip Muscarinic acetylcholine receptors | | Agonists |  | 
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 | Antagonists | 
- 3-Quinuclidinyl benzilate
 
- 4-DAMP
 
- Aclidinium bromide (+formoterol)
 
- Abediterol
 
- AF-DX 250
 
- AF-DX 384
 
- Ambutonium bromide
 
- Anisodamine
 
- Anisodine
 
- Antihistamines (first-generation) (e.g., brompheniramine, buclizine, captodiame, chlorphenamine (chlorpheniramine), cinnarizine, clemastine, cyproheptadine, dimenhydrinate, dimetindene, diphenhydramine, doxylamine, meclizine, mequitazine, perlapine, phenindamine, pheniramine, phenyltoloxamine, promethazine, propiomazine, triprolidine)
 
- AQ-RA 741
 
- Atropine
 
- Atropine methonitrate
 
- Atypical antipsychotics (e.g., clozapine, fluperlapine, olanzapine (+fluoxetine), rilapine, quetiapine, tenilapine, zotepine)
 
- Benactyzine
 
- Benzatropine (benztropine)
 
- Benzilone
 
- Benzilylcholine mustard
 
- Benzydamine
 
- Bevonium
 
- BIBN 99
 
- Biperiden
 
- Bornaprine
 
- Camylofin
 
- CAR-226,086
 
- CAR-301,060
 
- CAR-302,196
 
- CAR-302,282
 
- CAR-302,368
 
- CAR-302,537
 
- CAR-302,668
 
- Caramiphen
 
- Cimetropium bromide
 
- Clidinium bromide
 
- Cloperastine
 
- CS-27349
 
- Cyclobenzaprine
 
- Cyclopentolate
 
- Darifenacin
 
- DAU-5884
 
- Desfesoterodine
 
- Dexetimide
 
- DIBD
 
- Dicycloverine (dicyclomine)
 
- Dihexyverine
 
- Difemerine
 
- Diphemanil metilsulfate
 
- Ditran
 
- Drofenine
 
- EA-3167
 
- EA-3443
 
- EA-3580
 
- EA-3834
 
- Emepronium bromide
 
- Etanautine
 
- Etybenzatropine (ethybenztropine)
 
- Fenpiverinium
 
- Fentonium bromide
 
- Fesoterodine
 
- Flavoxate
 
- Glycopyrronium bromide (+beclometasone/formoterol, +indacaterol, +neostigmine)
 
- Hexahydrodifenidol
 
- Hexahydrosiladifenidol
 
- Hexbutinol
 
- Hexocyclium
 
- Himbacine
 
- HL-031,120
 
- Homatropine
 
- Imidafenacin
 
- Ipratropium bromide (+salbutamol)
 
- Isopropamide
 
- J-104,129
 
- Hyoscyamine
 
- Mamba toxin 3
 
- Mamba toxin 7
 
- Mazaticol
 
- Mebeverine
 
- Meladrazine
 
- Mepenzolate
 
- Methantheline
 
- Methoctramine
 
- Methylatropine
 
- Methylhomatropine
 
- Methylscopolamine
 
- Metixene
 
- Muscarinic toxin 7
 
- N-Ethyl-3-piperidyl benzilate
 
- N-Methyl-3-piperidyl benzilate
 
- Nefopam
 
- Octatropine methylbromide (anisotropine methylbromide)
 
- Orphenadrine
 
- Otenzepad (AF-DX 116)
 
- Otilonium bromide
 
- Oxapium iodide
 
- Oxitropium bromide
 
- Oxybutynin
 
- Oxyphencyclimine
 
- Oxyphenonium bromide
 
- PBID
 
- PD-102,807
 
- PD-0298029
 
- Penthienate
 
- Pethidine
 
- pFHHSiD
 
- Phenglutarimide
 
- Phenyltoloxamine
 
- Pipenzolate bromide
 
- Piperidolate
 
- Pirenzepine
 
- Piroheptine
 
- Pizotifen
 
- Poldine
 
- Pridinol
 
- Prifinium bromide
 
- Procyclidine
 
- Profenamine (ethopropazine)
 
- Propantheline bromide
 
- Propiverine
 
- Quinidine
 
- 3-Quinuclidinyl thiochromane-4-carboxylate
 
- Revefenacin
 
- Rociverine
 
- RU-47,213
 
- SCH-57,790
 
- SCH-72,788
 
- SCH-217,443
 
- Scopolamine (hyoscine)
 
- Scopolamine butylbromide (hyoscine butylbromide)
 
- Silahexacyclium
 
- Sofpironium bromide
 
- Solifenacin
 
- SSRIsTooltip Selective serotonin reuptake inhibitors (e.g., femoxetine, paroxetine)
 
- Telenzepine
 
- Terodiline
 
- Tetracyclic antidepressants (e.g., amoxapine, maprotiline, mianserin, mirtazapine)
 
- Tiemonium iodide
 
- Timepidium bromide
 
- Tiotropium bromide
 
- Tiquizium bromide
 
- Tofenacin
 
- Tolterodine
 
- Tricyclic antidepressants (e.g., amitriptyline (+perphenazine), amitriptylinoxide, butriptyline, cidoxepin, clomipramine, desipramine, desmethyldesipramine, dibenzepin, dosulepin (dothiepin), doxepin, imipramine, lofepramine, nitroxazepine, northiaden (desmethyldosulepin), nortriptyline, protriptyline, quinupramine, trimipramine)
 
- Tridihexethyl
 
- Trihexyphenidyl
 
- Trimebutine
 
- Tripitamine (tripitramine)
 
- Tropacine
 
- Tropatepine
 
- Tropicamide
 
- Tropine benzilate
 
- Trospium chloride
 
- Typical antipsychotics (e.g., chlorpromazine, chlorprothixene, cyamemazine (cyamepromazine), loxapine, mesoridazine, thioridazine)
 
- Umeclidinium bromide (+vilanterol)
 
- WIN-2299
 
- Xanomeline
 
- Zamifenacin
  
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 Precursors (and prodrugs) |  | 
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- See also
 
- Receptor/signaling modulators
 
- Nicotinic acetylcholine receptor modulators
 
- Acetylcholine metabolism/transport modulators
  
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 | 
|---|
 | nAChRsTooltip Nicotinic acetylcholine receptors | Agonists (and PAMsTooltip positive allosteric modulators) | 
- 5-HIAA
 
- 6-Chloronicotine
 
- A-84,543
 
- A-366,833
 
- A-582,941
 
- A-867,744
 
- ABT-202
 
- ABT-418
 
- ABT-560
 
- ABT-894
 
- Acetylcholine
 
- Altinicline
 
- Anabasine
 
- Anatabine
 
- Anatoxin-a
 
- AR-R17779
 
- Bephenium hydroxynaphthoate
 
- Butinoline
 
- Butyrylcholine
 
- Carbachol
 
- Choline
 
- Choline m-bromophenyl ether
 
- Cotinine
 
- Cytisine
 
- Decamethonium
 
- Desformylflustrabromine
 
- Dianicline
 
- Dimethylphenylpiperazinium
 
- Epibatidine
 
- Epiboxidine
 
- Ethanol (alcohol)
 
- Ethoxysebacylcholine
 
- EVP-4473
 
- EVP-6124
 
- Galantamine
 
- GTS-21
 
- Ispronicline
 
- Ivermectin
 
- JNJ-39393406
 
- Levamisole
 
- Lobeline
 
- MEM-63,908 (RG-3487)
 
- Morantel
 
- Nicotine (tobacco)
 
- NS-1738
 
- PHA-543,613
 
- PHA-709,829
 
- PNU-120,596
 
- PNU-282,987
 
- Pozanicline
 
- Pyrantel
 
- Rivanicline
 
- RJR-2429
 
- Sazetidine A
 
- SB-206553
 
- Sebacylcholine
 
- SIB-1508Y
 
- SIB-1553A
 
- SSR-180,711
 
- Suberyldicholine
 
- Suxamethonium (succinylcholine)
 
- Suxethonium (succinyldicholine)
 
- TC-1698
 
- TC-1734
 
- TC-1827
 
- TC-2216
 
- TC-5214
 
- TC-5619
 
- TC-6683
 
- Tebanicline
 
- Tribendimidine
 
- Tropisetron
 
- UB-165
 
- Varenicline
 
- WAY-317,538
 
- XY-4083
  
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 Antagonists (and NAMsTooltip negative allosteric modulators) |  | 
|---|
 
  | 
|---|
 Precursors (and prodrugs) |  | 
|---|
 
- See also
 
- Receptor/signaling modulators
 
- Muscarinic acetylcholine receptor modulators
 
- Acetylcholine metabolism/transport modulators
  
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