Receptor (ligands) | | GlyRTooltip Glycine receptor | 
- Positive modulators: Alcohols (e.g., brometone, chlorobutanol (chloretone), ethanol (alcohol), tert-butanol (2M2P), tribromoethanol, trichloroethanol, trifluoroethanol)
 
- Alkylbenzene sulfonate
 
- Anandamide
 
- Barbiturates (e.g., pentobarbital, sodium thiopental)
 
- Chlormethiazole
 
- D12-116
 
- Dihydropyridines (e.g., nicardipine)
 
- Etomidate
 
- Ginseng constituents (e.g., ginsenosides (e.g., ginsenoside-Rf))
 
- Glutamic acid (glutamate)
 
- Ivermectin
 
- Ketamine
 
- Neuroactive steroids (e.g., alfaxolone, pregnenolone (eltanolone), pregnenolone acetate, minaxolone, ORG-20599)
 
- Nitrous oxide
 
- Penicillin G
 
- Propofol
 
- Tamoxifen
 
- Tetrahydrocannabinol
 
- Triclofos
 
- Tropeines (e.g., atropine, bemesetron, cocaine, LY-278584, tropisetron, zatosetron)
 
- Volatiles/gases (e.g., chloral hydrate, chloroform, desflurane, diethyl ether (ether), enflurane, halothane, isoflurane, methoxyflurane, sevoflurane, toluene, trichloroethane (methyl chloroform), trichloroethylene)
 
- Xenon
 
- Zinc
  
- Antagonists: 2-Aminostrychnine
 
- 2-Nitrostrychnine
 
- 4-Phenyl-4-formyl-N-methylpiperidine
 
- αEMBTL
 
- Bicuculline
 
- Brucine
 
- Cacotheline
 
- Caffeine
 
- Colchicine
 
- Colubrine
 
- Cyanotriphenylborate
 
- Dendrobine
 
- Diaboline
 
- Endocannabinoids (e.g., 2-AG, anandamide (AEA))
 
- Gaboxadol (THIP)
 
- Gelsemine
 
- iso-THAZ
 
- Isobutyric acid
 
- Isonipecotic acid
 
- Isostrychnine
 
- Laudanosine
 
- N-Methylbicuculline
 
- N-Methylstrychnine
 
- N,N-Dimethylmuscimol
 
- Nipecotic acid
 
- Pitrazepin
 
- Pseudostrychnine
 
- Quinolines (e.g., 4-hydroxyquinoline, 4-hydroxyquinoline-3-carboxylic acid, 5,7-CIQA, 7-CIQ, 7-TFQ, 7-TFQA)
 
- RU-5135
 
- Sinomenine
 
- Strychnine
 
- Thiocolchicoside
 
- Tutin
  
- Negative modulators: Amiloride
 
- Benzodiazepines (e.g., bromazepam, clonazepam, diazepam, flunitrazepam, flurazepam)
 
- Corymine
 
- Cyanotriphenylborate
 
- Daidzein
 
- Dihydropyridines (e.g., nicardipine, nifedipine, nitrendipine)
 
- Furosemide
 
- Genistein
 
- Ginkgo constituents (e.g., bilobalide, ginkgolides (e.g., ginkgolide A, ginkgolide B, ginkgolide C, ginkgolide J, ginkgolide M))
 
- Imipramine
 
- NBQX
 
- Neuroactive steroids (e.g., 3α-androsterone sulfate, 3β-androsterone sulfate, deoxycorticosterone, DHEA sulfate, pregnenolone sulfate, progesterone)
 
- Opioids (e.g., codeine, dextromethorphan, dextrorphan, levomethadone, levorphanol, morphine, oripavine, pethidine, thebaine)
 
- Picrotoxin (i.e., picrotin and picrotoxinin)
 
- PMBA
 
- Riluzole
 
- Tropeines (e.g., bemesetron, LY-278584, tropisetron, zatosetron)
 
- Verapamil
 
- Zinc
  
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 | NMDARTooltip N-Methyl-D-aspartate receptor |  | 
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